Delavirdine


- TRADE NAME: Rescriptor (ViiV)
- INDICATIONS: HIV-1 infection
- CLASS: Antiretroviral, CYP3A4 inhibitor, Non-nucleoside reverse transcriptase inhibitor
- HALF-LIFE: 2–11 hours
Adefovir, Alfuzosin, Almotriptan, Alosetron, Alprazolam, Amiodarone, Amlodipine, Amphetamines, Amprenavir, Anisindione, Antacids, Anticoagulants, Artemether/Lumefantrine, Astemizole, Atomoxetine, Atorvastatin, Bepridil, Bortezomib, Brinzolamide, Buprenorphine, Carbamazepine, Carvedilol, Cerivastatin, Ciclesonide, Cimetidine, Cisapride, Clarithromycin, Clopidogrel, Codeine, Colchicine, Conivaptan, Cyclosporine, CYP2C19 substrates, CYP2C9 substrates, CYP2D6 substrates, CYP3A4 inducers and substrates, Darunavir, Deferasirox, Dexamethasone, Dicumarol, Dienogest, Dihydroergotamine, Diltiazem, Dronedarone, Dutasteride, Eplerenone, Ergonovine, Ergotamine, Estradiol, Etravirine, Everolimus, Famotidine, Felodipine, Fentanyl, Fesoterodine, Flecainide, Fluticasone Propionate, Fluvastatin, Fosamprenavir, Guanfacine, Halofantrine, Indinavir, Isradipine, Ixabepilone, Lansoprazole, Lidocaine, Lopinavir, Lovastatin, Maraviroc, Methadone, Methylergonovine, Methylprednisolone, Methysergide, Midazolam, Mometasone, Nebivolol, Nelfinavir, Nicardipine, Nifedipine, Nilotinib, Nimodipine, Nisoldipine, Nizatidine, Omeprazole, Paclitaxel, Pantoprazole, Paricalcitol, Pazopanib, PEG-Interferon, Phenobarbital, Phenytoin, Pimecrolimus, Pimozide, Prasugrel, Propafenone, Propranolol, Protease inhibitors, Proton pump inhibitors, Quinidine, Ranitidine, Ranolazine, Rifabutin, Rifampin, Rifapentine, Rilpivirine, Ritonavir, Rivaroxaban, Romidepsin, Salmeterol, Saquinavir, Saxagliptin, Sildenafil, Silodosin, Simeprevir, Simvastatin, Sirolimus, Sorafenib, St John's Wort, Tacrolimus, Tadalafil, Tamoxifen, Tamsulosin, Terfenadine, Tetrabenazine, Thioridazine, Tipranavir, Tolvaptan, Tramadol, Trazodone, Triazolam, Verapamil, Warfarin
PREGNANCY CATEGORY: C
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Page last updated 08/03/2022
Symbol key
Incidence 
- <1%
- 1-5%
- 5-10%
- 10-15%
- 15-20%
- 20-30%
- >30%
Warnings in other populations 
- Breast feeding
- Geriatric
- Pediatric