Pazopanib


- TRADE NAME: Votrient (Novartis)
- INDICATIONS: Advanced renal cell carcinoma
- CLASS: Angiogenesis inhibitor / antiangiogenic agent, Antineoplastic / anticancer agent (see also Immune checkpoint inhibitor), Tyrosine kinase inhibitor, Vascular endothelial growth factor (VEGF) inhibitor / antagonist
- HALF-LIFE: 31 hours
Alfuzosin, Artemether/Lumefantrine, Atazanavir, BCG Vaccine, Boceprevir, Cardiac glycosides, Chloroquine, Ciprofloxacin, Clarithromycin, Clozapine, Conivaptan, CYP3A4 inducers or inhibitors, Cyproterone, Darunavir, Deferasirox, Delavirdine, Denosumab, Dronedarone, Efavirenz, Gadobutrol, Grapefruit Juice, Indacaterol, Indinavir, Itraconazole, Ketoconazole, Lapatinib, Leflunomide, Natalizumab, Nelfinavir, Nilotinib, Oxcarbazepine, P-glycoprotein inhibitors, Pimecrolimus, Pimozide, QT prolonging agents, Quetiapine, Quinine, Rifampin, Rifapentine, Ritonavir, Roflumilast, Saquinavir, Simvastatin, Sipuleucel-T, St John's Wort, Tacrolimus, Telithromycin, Tetrabenazine, Thioridazine, Tocilizumab, Toremifene, Trastuzumab, Vaccines, Vandetanib, Vemurafenib, Vitamin K antagonists, Voriconazole, Ziprasidone
PREGNANCY CATEGORY: D
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Page last updated 08/03/2023
Symbol key
Incidence 
- <1%
- 1-5%
- 5-10%
- 10-15%
- 15-20%
- 20-30%
- >30%
Warnings in other populations 
- Breast feeding
- Geriatric
- Pediatric