Conivaptan


- TRADE NAME: Vaprisol (Astellas)
- INDICATIONS: Hyponatremia, SIADH
- CLASS: CYP3A4 inhibitor, Vasopressin receptor antagonist
- HALF-LIFE: 5 hours
Acetaminophen, Albendazole, Alfuzosin, Almotriptan, Alosetron, Ambrisentan, Amitriptyline, Amlodipine, Antifungals, Aprepitant, Artemether/Lumefantrine, Atorvastatin, Bexarotene, Bortezomib, Brigatinib, Brinzolamide, Bupivacaine, Cabazitaxel, Cabozantinib, Ciclesonide, Cilostazol, Cinacalcet, Citalopram, Clarithromycin, Colchicine, Copanlisib, Cyclobenzaprine, CYP3A4 inhibitors or substrates, Darunavir, Dasatinib, Deferasirox, Delavirdine, Dienogest, Digoxin, Docetaxel, Dolasetron, Dronedarone, Dutasteride, Efavirenz, Enalapril, Eplerenone, Estradiol, Eszopiclone, Everolimus, Fentanyl, Fesoterodine, Fingolimod, Flibanserin, Gefitinib, Guanfacine, Halofantrine, Indinavir, Itraconazole, Ixabepilone, Ketoconazole, Lapatinib, Lomitapide, Maraviroc, Meloxicam, Metaxalone, Methylprednisolone, Micafungin, Midazolam, Midostaurin, Mifepristone, Mometasone, Neratinib, Nilotinib, Nisoldipine, Oxybutynin, Pantoprazole, Paricalcitol, Pazopanib, Pimecrolimus, Pioglitazone, Ponatinib, Prasugrel, Ramelteon, Ranolazine, Ribociclib, Ritonavir, Rivaroxaban, Romidepsin, Rosuvastatin, Ruxolitinib, Salmeterol, Saxagliptin, Sildenafil, Silodosin, Simvastatin, Sorafenib, St John's Wort, Tadalafil, Tamsulosin, Telithromycin, Temsirolimus, Terbinafine, Tiagabine, Tiotropium, Tipranavir, Tolvaptan, Trimethoprim, Ulipristal, Vardenafil, Venetoclax, Vorapaxar, Voriconazole, Ziprasidone
PREGNANCY CATEGORY: C
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Page last updated 07/31/2023
Symbol key
Incidence 
- <1%
- 1-5%
- 5-10%
- 10-15%
- 15-20%
- 20-30%
- >30%
Warnings in other populations 
- Breast feeding
- Geriatric
- Pediatric