Darunavir


- TRADE NAMES: Prezcobix (Janssen); Prezista (Janssen)
- INDICATIONS: HIV infection (must be co-administered with ritonavir and with other antiretroviral agents)
- CLASS: Antiretroviral, Covid-19 putative drug, HIV-1 protease inhibitor
- HALF-LIFE: 15 hours
Abacavir, Alfuzosin, Almotriptan, Alosetron, Alprazolam, Amiodarone, Antifungals, Apixaban, Artemether/Lumefantrine, Astemizole, Atorvastatin, Bortezomib, Brinzolamide, Calcium channel blockers, Captopril, Carbamazepine, Ciclesonide, Cisapride, Clarithromycin, Colchicine, Conivaptan, Cyclosporine, CYP2D6 substrates, CYP3A4 inhibitors, inducers and substrates, Dabigatran, Dasatinib, Deferasirox, Delavirdine, Didanosine, Dienogest, Digoxin, Dihydroergotamine, Dronedarone, Duloxetine, Dutasteride, Efavirenz, Elbasvir & Grazoprevir, Enfuvirtide, Eplerenone, Ergotamine, Estrogens, Etravirine, Everolimus, Fentanyl, Fesoterodine, Food, Fusidic Acid, Glecaprevir & Pibrentasvir, Guanfacine, Halofantrine, HMG-CoA reductase inhibitors, Indinavir, Inhaled corticosteroids, Ixabepilone, Ketoconazole, Lidocaine, Lopinavir, Lovastatin, Maraviroc, Meperidine, Methadone, Methylprednisolone, Midazolam, Mifepristone, Mometasone, Nefazodone, Nilotinib, Nisoldipine, Olaparib, P-glycoprotein substrates, Paricalcitol, Paroxetine Hydrochloride, Pazopanib, Phenobarbital, Phenytoin, Pimecrolimus, Pimozide, Prasugrel, Pravastatin, Protease inhibitors, Quetiapine, Quinidine, Quinine, Ranolazine, Rifabutin, Rifampin, Rilpivirine, Rivaroxaban, Romidepsin, Rosuvastatin, Salmeterol, Saquinavir, Saxagliptin, Sertraline, Sildenafil, Silodosin, Simeprevir, Simvastatin, Sirolimus, Sorafenib, St John's Wort, Tacrolimus, Tadalafil, Tamsulosin, Telaprevir, Temsirolimus, Tenofovir Disoproxil, Terfenadine, Theophylline, Tolvaptan, Topotecan, Trazodone, Triazolam, Tricyclic antidepressants, Vardenafil, Viloxazine, Voriconazole, Warfarin, Zidovudine
PREGNANCY CATEGORY: C
Investigated for treating COVID-19.
Darunavir is a sulfonamide and can be absorbed systemically. Sulfonamides can produce severe, possibly fatal, reactions such as toxic epidermal necrolysis and Stevens-Johnson syndrome.
Prezcobix is darunavir and cobicistat.
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Page last updated 07/31/2023
Symbol key
Incidence 
- <1%
- 1-5%
- 5-10%
- 10-15%
- 15-20%
- 20-30%
- >30%
Warnings in other populations 
- Breast feeding
- Geriatric
- Pediatric