Amprenavir


- TRADE NAME: Agenerase (GSK)
- INDICATIONS: HIV infection
- CLASS: Antiretroviral, HIV-1 protease inhibitor
- HALF-LIFE: 7–11 hours
Alprazolam, Amiodarone, Amitriptyline, Amlodipine, Amoxapine, Antacids, Atorvastatin, Avanafil, Benzodiazepines, Bepridil, Bosentan, Carbamazepine, Cisapride, Clomipramine, Clonazepam, Clorazepate, Cyclosporine, Delavirdine, Desipramine, Dexamethasone, Diazepam, Didanosine, Dihydroergotamine, Diltiazem, Doxepin, Efavirenz, Ergotamine, Estradiol, Felodipine, Fentanyl, Flibanserin, Flurazepam, Fluticasone Propionate, Imipramine, Indinavir, Isradipine, Itraconazole, Ixabepilone, Ketoconazole, Lidocaine, Lopinavir, Lorazepam, Lovastatin, Lumateperone, Methadone, Methylergonovine, Methysergide, Midazolam, Mifepristone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldipine, Nortriptyline, Olaparib, Oral Contraceptives, Oxazepam, Phenobarbital, Phenytoin, Pimozide, Protriptyline, Quazepam, Quinidine, Rapamycin, Rifabutin, Rifampin, Ritonavir, Saquinavir, Sildenafil, Simvastatin, St John's Wort, Tacrolimus, Temazepam, Trazodone, Triazolam, Tricyclic antidepressants, Trimipramine, Verapamil, Vitamin E, Warfarin
PREGNANCY CATEGORY: C
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Page last updated 08/01/2022
Symbol key
Incidence 
- <1%
- 1-5%
- 5-10%
- 10-15%
- 15-20%
- 20-30%
- >30%
Warnings in other populations 
- Breast feeding
- Geriatric
- Pediatric