Amprenavir


- TRADE NAME: Agenerase (GSK)
- INDICATIONS: HIV infection
- CLASS: Antiretroviral, HIV-1 protease inhibitor
- HALF-LIFE: 7–11 hours
Alprazolam, Amiodarone, Amitriptyline, Amlodipine, Amoxapine, Antacids, Atorvastatin, Avanafil, Benzodiazepines, Bepridil, Bosentan, Carbamazepine, Cisapride, Clomipramine, Clonazepam, Clorazepate, Cyclosporine, Delavirdine, Desipramine, Dexamethasone, Diazepam, Didanosine, Dihydroergotamine, Diltiazem, Doxepin, Efavirenz, Ergotamine, Estradiol, Felodipine, Fentanyl, Flibanserin, Flurazepam, Fluticasone Propionate, Imipramine, Indinavir, Isradipine, Itraconazole, Ixabepilone, Ketoconazole, Lidocaine, Lopinavir, Lorazepam, Lovastatin, Lumateperone, Methadone, Methylergonovine, Methysergide, Midazolam, Mifepristone, Nelfinavir, Nevirapine, Nicardipine, Nifedipine, Nimodipine, Nisoldipine, Nortriptyline, Olaparib, Oral Contraceptives, Oxazepam, Phenobarbital, Phenytoin, Pimozide, Protriptyline, Quazepam, Quinidine, Rapamycin, Rifabutin, Rifampin, Ritonavir, Saquinavir, Sildenafil, Simvastatin, St John's Wort, Tacrolimus, Temazepam, Trazodone, Triazolam, Tricyclic antidepressants, Trimipramine, Verapamil, Vitamin E, Warfarin
PREGNANCY CATEGORY: C
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Page last updated 07/31/2023
Symbol key
Incidence 
- <1%
- 1-5%
- 5-10%
- 10-15%
- 15-20%
- 20-30%
- >30%
Warnings in other populations 
- Breast feeding
- Geriatric
- Pediatric