Cobicistat/Elvitegravir/Emtricitabine/Tenofovir Alafenamide

- TRADE NAME: Genvoya (Gilead)
- INDICATIONS: HIV-1 infection
- CLASS: Antiretroviral, CYP3A inhibitor (cobicistat), Hepatitis B virus necleoside analog reverse transcriptase inhibitor (tenofovir alafenamide), Integrase strand transfer inhibitor (elvitegravir), Nucleoside analog reverse transcriptase inhibitor (emtricitabine)
- HALF-LIFE: 3.5 hours (cobicistat); 13 hours (elvitegravir); 10 hours (emtricitabine); <1 hour (tenofovir alafenamide)
FDA APPROVAL DATE: 11/05/2015 (Genvoya)
CLINICALLY IMPORTANT, POTENTIALLY HAZARDOUS INTERACTIONS WITH:Acyclovir, Aminoglycosides, Amiodarone, Amitriptyline, Amlodipine, Antacids, Antiarrhythmics, Atorvastatin, Benzodiazepines, Bepridil, Beta blockers, Bosentan, Buprenorphine, Bupropion, Buspirone, Calcium channel blockers, Cidofovir, Clarithromycin, Clorazepate, Colchicine, Desipramine, Dexamethasone, Diazepam, Digoxin, Diltiazem, Disopyramide, Drugs affecting renal function, Estazolam, Ethosuximide, Felodipine, Flecainide, Flurazepam, Fluticasone Furoate, Fluticasone Propionate, Ganciclovir, Gentamicin, Hormonal contraceptives, Imipramine, Immunosuppressants, Itraconazole, Ketoconazole, Lidocaine, Lorazepam, Metoprolol, Mexiletine, Midazolam, Naloxone, Neuroleptics, Nicardipine, Nifedipine, Nortriptyline, Oxcarbazepine, Paroxetine Hydrochloride, Perphenazine, Propafenone, Quinidine, Rifabutin, Rifapentine, Risperidone, Salmeterol, Sildenafil, SSRIs, Tadalafil, Telithromycin, Thioridazine, Timolol, Trazodone, Tricyclic antidepressants, Valacyclovir, Valganciclovir, Vardenafil, Verapamil, Voriconazole, Warfarin, Zolpidem
PREGNANCY CATEGORY: B
See also separate profiles for emtricitabine and tenofovir alafenamide.
See full prescribing information for complete boxed warning.
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Page last updated 08/03/2022
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Incidence 
- <1%
- 1-5%
- 5-10%
- 10-15%
- 15-20%
- 20-30%
- >30%
Warnings in other populations 
- Breast feeding
- Geriatric
- Pediatric