Sunitinib


- TRADE NAME: Sutent (Pfizer)
- INDICATIONS: Gastrointestinal stromal tumor, advanced renal cell carcinoma, advanced pancreatic neuroendocrine tumor
- CLASS: Antineoplastic / anticancer agent (see also Immune checkpoint inhibitor), Tyrosine kinase inhibitor, Vascular endothelial growth factor (VEGF) inhibitor / antagonist
- HALF-LIFE: 40–60 hours
Atazanavir, Bevacizumab, Carbamazepine, Clarithromycin, Clozapine, Dexamethasone, Digoxin, Efavirenz, Grapefruit Juice, Indinavir, Itraconazole, Ketoconazole, Nefazodone, Nelfinavir, Phenobarbital, Phenytoin, Rifabutin, Rifampin, Rifapentine, Ritonavir, Saquinavir, St John's Wort, Telithromycin, Temsirolimus, Voriconazole
PREGNANCY CATEGORY: D
[G] = treated for gastrointestinal tumor; [R] = treated for renal cell carcinoma; [P] treated for pancreatic neuroendocrine tumor
See full prescribing information for complete boxed warning.
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Page last updated 04/05/2023
Symbol key
Incidence 
- <1%
- 1-5%
- 5-10%
- 10-15%
- 15-20%
- 20-30%
- >30%
Warnings in other populations 
- Breast feeding
- Geriatric
- Pediatric