Litt’s Drug profile for Relugolix

  • FDA Approval Date: 12/18/2020
  • Clinically important, potentially hazardous interactions with:
    CYP3A inducers, Erythromycin, P-gp inhibitors, Rifampin
  • Pregnancy: Relugolix can cause fetal harm. Advise males with female partners of reproductive potential to use effective contraception.

Androgen deprivation therapy, such as Relugolix, may prolong the QT/QTc interval.

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Page last updated 09/25/2026

Symbol key

Incidence - Help

<1% 1‑5% 5‑10% 10‑15% 15‑20% 20‑30% >30%

Seriousness - Help

Hospitalization possible
Life threatening
Fatal

Warnings in other populations - Help

BreastfeedingBreast feeding

GeriatricGeriatric

PediatricPediatric