Telaprevir
- TRADE NAME: Incivek (Vertex)
- INDICATIONS: Hepatitis C (must only be used in combination with PEG-interferon alfa and ribavirin)
- CLASS: CYP3A4 inhibitor, Direct-acting antiviral, Hepatitis C virus NS3/4A protease inhibitor
- HALF-LIFE: 4–11 hours
Alfuzosin, Alprazolam, Amiodarone, Amlodipine, Atazanavir, Atorvastatin, Bepridil, Bosentan, Budesonide, Carbamazepine, Cisapride, Dabigatran, Darunavir, Desipramine, Dexamethasone, Digoxin, Dihydroergotamine, Diltiazem, Efavirenz, Ergotamine, Escitalopram, Estradiol, Felodipine, Flecainide, Flibanserin, Fluticasone Propionate, Fosamprenavir, Itraconazole, Ketoconazole, Lidocaine, Lomitapide, Lovastatin, Methylergonovine, Methylprednisolone, Midazolam, Mifepristone, Nicardipine, Nisoldipine, Olaparib, Palbociclib, Phenobarbital, Phenytoin, Pimozide, Ponatinib, Posaconazole, Propafenone, Quinidine, Rifampin, Ritonavir, Ruxolitinib, Salmeterol, Sildenafil, Simvastatin, Sirolimus, St John's Wort, Tacrolimus, Tadalafil, Telithromycin, Tenofovir Disoproxil, Trazodone, Triazolam, Vardenafil, Venetoclax, Verapamil, Vorapaxar, Voriconazole, Warfarin, Zolpidem
PREGNANCY CATEGORY: X
Must be used in combination with PEG-interferon alfa and ribavirin (see separate entries)
See full prescribing information for complete boxed warning.
Please login to see the rest of this drug profile
Page last updated 07/31/2023
Symbol key
Incidence
- <1%
- 1-5%
- 5-10%
- 10-15%
- 15-20%
- 20-30%
- >30%
Warnings in other populations
- Breast feeding
- Geriatric
- Pediatric